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dc.contributor.authorChakrabarty, Manas
dc.contributor.authorKundu, Taraknath
dc.contributor.authorArima, S.
dc.contributor.authorHarigaya, Y.
dc.date.accessioned2013-04-02T07:23:56Z
dc.date.available2013-04-02T07:23:56Z
dc.date.issued2005-04-18
dc.identifierFOR ACCESS / DOWNLOAD PROBLEM -- PLEASE CONTACT LIBRARIAN, BOSE INSTITUTE, akc@bic.boseinst.ernet.inen_US
dc.identifier.citationChakrabarty M, Kundu T, Arima S and Harigaya Y (2005) An expedient, regioselective synthesis of 2-alkylamino- and 2-alkylthiothiazolo[5,4-e ]indoles. Tetrahedron Lett. 44 (16), 2865-2868.en_US
dc.identifier.issn0040-4039
dc.identifier.uri1.Full Text Link ->
dc.identifier.urihttp://ac.els-cdn.com/S004040390500434X/1-s2.0-S004040390500434X-main.pdf?_tid=d0175a92-9b65-11e2-a330-00000aab0f27&acdnat=1364887416_d4a532ca0baa924d4a7da538a71077a5en_US
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dc.identifier.uri2. Scopus : Citation Link ->en_US
dc.identifier.urihttp://www.scopus.com/record/display.url?eid=2-s2.0-15944381575&origin=resultslist&sort=plf-f&src=s&nlo=&nlr=&nls=&sid=DEE7BF283ED6E12BE230003963403DAE.N5T5nM1aaTEF8rE6yKCR3A%3a30&sot=aut&sdt=a&sl=38&s=AU-ID%28%22Chakrabarty%2c+Manas%22+7006688171%29&relpos=19&relpos=19&searchTerm=AU-ID%28\%26quot%3BChakrabarty%2C+Manas\%26quot%3B+7006688171%29en_US
dc.descriptionDOI: 10.1016/j.tetlet.2005.02.125en_US
dc.description.abstract1-Benzenesulfonyl-5-aminoindole 5, prepared from 5-nitroindole 3, was condensed with alkyl isothiocyanates and separately with carbon disulfide and alkyl bromides/iodides to furnish efficiently the corresponding N-alkyl-thioureidoindoles 6a-c and the alkyl N'-(indol-5'-yl)dithiocarbamates 9a-e, respectively. Their cyclisation using N-bromosuccinimide (NBS) and 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU), in the cold, followed by indolic N-deprotection, furnished regioselectively the 2-alkylamino- and the 2-alkylthiothiazolo[5,4-e]indoles 8a-c and 11a-e, respectively, in good overall yields.en_US
dc.language.isoenen_US
dc.publisherPERGAMON-ELSEVIER SCIENCE LTDen_US
dc.subjectthiazolo[5,4-e]indolesen_US
dc.subjectregioselective synthesisen_US
dc.subjectthioureido-indolesen_US
dc.subjectindolyldithiocarbamatesen_US
dc.subjectNBS-DBUen_US
dc.subjectANR-2005-06en_US
dc.titleAn expedient, regioselective synthesis of 2-alkylamino- and 2-alkylthiothiazolo[5,4-e]indolesen_US
dc.title.alternativeTetrahedron Lettersen_US
dc.typeArticleen_US


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