| dc.contributor.author | Chakrabarty, Manas | |
| dc.contributor.author | Kundu, Taraknath | |
| dc.contributor.author | Arima, S. | |
| dc.contributor.author | Harigaya, Y. | |
| dc.date.accessioned | 2013-04-02T07:23:56Z | |
| dc.date.available | 2013-04-02T07:23:56Z | |
| dc.date.issued | 2005-04-18 | |
| dc.identifier | FOR ACCESS / DOWNLOAD PROBLEM -- PLEASE CONTACT LIBRARIAN, BOSE INSTITUTE, akc@bic.boseinst.ernet.in | en_US |
| dc.identifier.citation | Chakrabarty M, Kundu T, Arima S and Harigaya Y (2005) An expedient, regioselective synthesis of 2-alkylamino- and 2-alkylthiothiazolo[5,4-e ]indoles. Tetrahedron Lett. 44 (16), 2865-2868. | en_US |
| dc.identifier.issn | 0040-4039 | |
| dc.identifier.uri | 1.Full Text Link -> | |
| dc.identifier.uri | http://ac.els-cdn.com/S004040390500434X/1-s2.0-S004040390500434X-main.pdf?_tid=d0175a92-9b65-11e2-a330-00000aab0f27&acdnat=1364887416_d4a532ca0baa924d4a7da538a71077a5 | en_US |
| dc.identifier.uri | ================================================= | en_US |
| dc.identifier.uri | 2. Scopus : Citation Link -> | en_US |
| dc.identifier.uri | http://www.scopus.com/record/display.url?eid=2-s2.0-15944381575&origin=resultslist&sort=plf-f&src=s&nlo=&nlr=&nls=&sid=DEE7BF283ED6E12BE230003963403DAE.N5T5nM1aaTEF8rE6yKCR3A%3a30&sot=aut&sdt=a&sl=38&s=AU-ID%28%22Chakrabarty%2c+Manas%22+7006688171%29&relpos=19&relpos=19&searchTerm=AU-ID%28\%26quot%3BChakrabarty%2C+Manas\%26quot%3B+7006688171%29 | en_US |
| dc.description | DOI: 10.1016/j.tetlet.2005.02.125 | en_US |
| dc.description.abstract | 1-Benzenesulfonyl-5-aminoindole 5, prepared from 5-nitroindole 3, was condensed with alkyl isothiocyanates and separately with carbon disulfide and alkyl bromides/iodides to furnish efficiently the corresponding N-alkyl-thioureidoindoles 6a-c and the alkyl N'-(indol-5'-yl)dithiocarbamates 9a-e, respectively. Their cyclisation using N-bromosuccinimide (NBS) and 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU), in the cold, followed by indolic N-deprotection, furnished regioselectively the 2-alkylamino- and the 2-alkylthiothiazolo[5,4-e]indoles 8a-c and 11a-e, respectively, in good overall yields. | en_US |
| dc.language.iso | en | en_US |
| dc.publisher | PERGAMON-ELSEVIER SCIENCE LTD | en_US |
| dc.subject | thiazolo[5,4-e]indoles | en_US |
| dc.subject | regioselective synthesis | en_US |
| dc.subject | thioureido-indoles | en_US |
| dc.subject | indolyldithiocarbamates | en_US |
| dc.subject | NBS-DBU | en_US |
| dc.subject | ANR-2005-06 | en_US |
| dc.title | An expedient, regioselective synthesis of 2-alkylamino- and 2-alkylthiothiazolo[5,4-e]indoles | en_US |
| dc.title.alternative | Tetrahedron Letters | en_US |
| dc.type | Article | en_US |